Bromocriptine mesylate
Bromocriptine mesylate
Bromocriptine mesylate
| Catalog | Description | Size | Price (USD) | Qty |
|---|---|---|---|---|
| GBM-1096-100MG | Bromocriptine mesylate | 100mg | $137.00 | |
| GBM-1096-500MG | Bromocriptine mesylate | 500mg | $546.00 |
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Description
Dopamine D2/D3 agonist
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Specifications
Bioassays Specification Bio-Activity Dopamine D2/D3 agonist Chemical Name (+)-2-Bromo-12’-hydroxy-2’-(1-methylethyl)-5’-(2-methylpropyl)-ergotaman-3’,6,’18-trione methanesulfonate Function / Pharmacology Dopamine D2 receptor agonist. Inhibits prolactin production3. Decreases cocaine self-administration in the rat4. Active in vivo. CAS# 22260-51-1 MW 750.7 Molecular Formula C32H40BrN5O5 • CH3SO3H Solubility Soluble in DMSO (up to 50 mg/ml) or in Ethanol (up to 6 mg/ml). Supplied powder Storage as supplied RT Ship temp Ambient References 1) Nilsson and Hokfelt (1978), Effect of the dopamine agonist bromocriptine on blood pressure, catecholamines and renin activity in acromegalics at rest, following exercise, and during insulin induced hypoglycemia; Acta Endocrinol., Supp. 216 83 2) Seeman and Van Tol (1994), Dopamine receptor pharmacology; Trends Pharmacol. Sci., 15 264 3) Carvalho et al. (2015), Maternal prolactin inhibition causes changes in leptin at 22- and 30-day old pups; Horm. Metab. Res., 47 528 4) Hubner and Koob (1990), Bromocriptine produces decreases in cocaine self-administration in the rat; Neuropsychopharmacol., 3 101 Protein Specification Purity >98% - Reviews
| Bioassays Specification | |
| Bio-Activity | Dopamine D2/D3 agonist |
| Chemical Name | (+)-2-Bromo-12’-hydroxy-2’-(1-methylethyl)-5’-(2-methylpropyl)-ergotaman-3’,6,’18-trione methanesulfonate |
| Function / Pharmacology | Dopamine D2 receptor agonist. Inhibits prolactin production3. Decreases cocaine self-administration in the rat4. Active in vivo. |
| CAS# | 22260-51-1 |
| MW | 750.7 |
| Molecular Formula | C32H40BrN5O5 • CH3SO3H |
| Solubility | Soluble in DMSO (up to 50 mg/ml) or in Ethanol (up to 6 mg/ml). |
| Supplied | powder |
| Storage as supplied | RT |
| Ship temp | Ambient |
| References | 1) Nilsson and Hokfelt (1978), Effect of the dopamine agonist bromocriptine on blood pressure, catecholamines and renin activity in acromegalics at rest, following exercise, and during insulin induced hypoglycemia; Acta Endocrinol., Supp. 216 83 2) Seeman and Van Tol (1994), Dopamine receptor pharmacology; Trends Pharmacol. Sci., 15 264 3) Carvalho et al. (2015), Maternal prolactin inhibition causes changes in leptin at 22- and 30-day old pups; Horm. Metab. Res., 47 528 4) Hubner and Koob (1990), Bromocriptine produces decreases in cocaine self-administration in the rat; Neuropsychopharmacol., 3 101 |
| Protein Specification | |
| Purity | >98% |